Imidafenacin

Catalog No.: A15490

M3 receptors inhibitor

Imidafenacin

Imidafenacin Chemical Structure

CAS NO. 170105-16-5

Imidafenacin is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors(IC50=4.13 nM).

Availability: In stock

Package Price Qty
10 mg
$45.00
25 mg
$90.00
50 mg
$155.00
100 mg
$265.00
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Biological Activity

Imidafenacin is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors(IC50=4.13 nM).
In vitro DMSO 60 mg/mL (187.85 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 31.31 mL 156.54 mL 313.09 mL
0.5 mM 6.26 mL 31.31 mL 62.62 mL
1 mM 3.13 mL 15.65 mL 31.31 mL
5 mM 0.63 mL 3.13 mL 6.26 mL

*The above data is based on the productmolecular weight 319.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15490
Actions Inhibitor
CAS No. 170105-16-5
Formula C20H21N3O
M. Wt 319.4
Solubility DMSO
Purity >98%
Synonyms KRP-197, ONO-8025
SMILES CC1=NC=CN1CCC(C2=CC=CC=C2)(C3=CC=CC=C3)C(=O)N
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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