Fig. 1 · Structure
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IP3RPEP6
IP3R Inhibitor
IP3RPEP6 is a competitive inhibitor of inositol trisphosphate receptors (IP3R), demonstrating IC50 values of 9.0 μM, 3.9 μM, and 4.3 μM for IP3R1, IP3R2, and IP3R3, respectively. This compound selectively targets IP3 receptors without influencing ryanodine receptors or connexin 43 hemichannels. IP3RPEP6 plays a crucial role in modulating intracellular calcium signaling, making it a valuable tool for research focused on cellular calcium dynamics and related signaling pathways.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 3061802-23-8 |
| Applications | IP3R Inhibitor |
| Formula | C49H79N15O24 |
| Molecular Weight | 1262.24 |
| SMILES | [C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC(N)=O)C(O)=O)=O)CO)=O)CCC(O)=O)=O)(NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC(CNC(CNC([C@@H](NC([C@H](C(C)C)N)=O)CCCCN)=O)=O)=O)CCC(O)=O)=O)CCC(O)=O)=O)C)=O)CC(N)=O)=O)CCC(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.