Fig. 1 · Structure
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JG-2016
HAT1 Inhibitor
JG-2016 is a potent inhibitor of histone acetyltransferase 1 (HAT1), exhibiting an IC50 of 14.8 μM. This compound effectively suppresses the growth of various tumor cell lines and demonstrates significant anti-tumor activity. JG-2016 is valuable for research applications focused on cancer biology and epigenetic regulation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2887480-87-5 |
| Applications | HAT1 Inhibitor |
| Formula | C18H21ClN4O3 |
| Molecular Weight | 376.84 |
| SMILES | O=C(N1)N=C2N(CCOCC(C)C)C3=CC(CC)=C(Cl)C=C3N=C2C1=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.