JNJ-17203212

Catalog No.: A12766

TRPV1 antagonist

JNJ-17203212

JNJ-17203212 Chemical Structure

CAS NO. 821768-06-3

NJ-17203212 is a novel and selective TRPV1 antagonist, with IC50 of 65 nM and 102 nM for human TRPV1 and rat TRPV1.

Availability: In stock

Package Price Qty
5 mg
$81.00
10 mg
$140.00
50 mg
$414.00
100 mg
$828.00
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Biological Activity

NJ-17203212 is a novel and selective TRPV1 antagonist, with IC50 of 65 nM and 102 nM for human TRPV1 and rat TRPV1.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.85 mL 119.24 mL 238.48 mL
0.5 mM 4.77 mL 23.85 mL 47.7 mL
1 mM 2.38 mL 11.92 mL 23.85 mL
5 mM 0.48 mL 2.38 mL 4.77 mL

*The above data is based on the productmolecular weight 419.32. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12766
Actions Antagonist
CAS No. 821768-06-3
Formula C17H15F6N5O
M. Wt 419.32
Solubility DMSO
Purity >98%
Synonyms JNJ17203212, JNJ 17203212
SMILES O=C(N1CCN(C2=NC=CC=C2C(F)(F)F)CC1)NC3=NC=C(C(F)(F)F)C=C3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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