L-R4W2

Name: L-R4W2
Brand: Adooq Bioscience
SKU: A68771
Rating: 5 (288 reviews)

Catalog No.: A68771

TRPV1 Antagonist

L-R4W2 is a potent antagonist of the vanilloid receptor 1 (VR1, TRPV1), exhibiting an IC50 of 0.1 μM. This compound demonstrates significant analgesic properties, making it a valuable tool in pain management research. L-R4W2 can be utilized to explore mechanisms of pain signaling and the therapeutic potential for treating pain-related disorders.

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Size	Price	Stock	Qty
1mg	$180.00	In stock
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Biological Activity

Description	L-R4W2 is a potent antagonist of the vanilloid receptor 1 (VR1, TRPV1), exhibiting an IC50 of 0.1 μM. This compound demonstrates significant analgesic properties, making it a valuable tool in pain management research. L-R4W2 can be utilized to explore mechanisms of pain signaling and the therapeutic potential for treating pain-related disorders.

Product Information

Catalog Num	A68771
Formula	C46H71N21O6
Molecular Weight	1014.19
CAS Number	206350-79-0
Sequence	Arg-Arg-Arg-Arg-Trp-Trp-NH2
Sequence shortening	RRRRWW-NH2
SMILES	C([C@@H](C(N[C@@H](CC=1C=2C(NC1)=CC=CC2)C(N)=O)=O)NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CCCNC(=N)N)N)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)C=3C=4C(NC3)=CC=CC4

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