Lanraplenib

Catalog No.: A12959

SYK inhibitor

Lanraplenib

Lanraplenib Chemical Structure

CAS NO. 1800046-95-0

Lanraplenib (GS-9876) is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases.

Availability: In stock

Package Price Qty
5 mg
$113.00
10 mg
$192.00
50 mg
$565.00
100 mg
$1,921.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Lanraplenib (GS-9876) is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases.
In vitro DMSO 77 mg/mL (173.61 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.55 mL 112.74 mL 225.48 mL
0.5 mM 4.51 mL 22.55 mL 45.1 mL
1 mM 2.25 mL 11.27 mL 22.55 mL
5 mM 0.45 mL 2.25 mL 4.51 mL

*The above data is based on the productmolecular weight 443.5. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12959
Actions Inhibitor
CAS No. 1800046-95-0
Formula C23H25N9O
M. Wt 443.5
Solubility DMSO
Purity >98%
Synonyms GS-9876, GS9876, GS 9876
SMILES NC1=CN=CC(C2=CN3C(C(NC4=CC=C(N5CCN(C6COC6)CC5)C=C4)=N2)=NC=C3)=N1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Lanraplenib | Lanraplenib Supplier | purchase | cost | manufacturer | order | distributor | buy 1800046-95-0| 1800046-95-0 Supplier | purchase 1800046-95-0 | 1800046-95-0 cost | 1800046-95-0 manufacturer | order 1800046-95-0 | 1800046-95-0 distributor
Rewards