Documents & Downloads

LDHA-IN-9

LDHA Inhibitor

LDHA-IN-9 is a potent lactate dehydrogenase A (LDHA) inhibitor, exhibiting an IC50 of 25 nM. This compound effectively inhibits DLD-1 cell proliferation with a GI50 of 27 μM, primarily by inducing apoptosis. Additionally, LDHA-IN-9 demonstrates significant antitumor activity in murine models while maintaining a favorable toxicity profile at a dosage of 25 mg/kg. This compound is suitable for research applications targeting metabolic regulation and cancer therapeutics.

Out of Stock

Free Aliquoting for Your Order

Tell us your preferred amount per vial. We’ll confirm the options.

Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	862719-04-8
Applications	LDHA Inhibitor
Formula	C₁₇H₂₂BrNO₄
Molecular Weight	384.26
SMILES	BrC1=C2C(N(O)C(C(OC)=O)=C2COCCCCCC)=CC=C1

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.