Fig. 1 · Structure
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LDN-209929
Haspin Inhibitor
LDN-209929 is a highly selective inhibitor of the haspin kinase, displaying an IC50 value of 55 nM for Haspin and 9.9 μM for DYRK2. This compound is utilized in research exploring the regulation of mitosis and cell division by specifically targeting the phosphorylation of histone H3. LDN-209929 serves as a valuable tool for investigating cancer biology and the mechanisms underlying various cell cycle-related processes.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1233355-57-1 |
| Applications | Haspin Inhibitor |
| Formula | C17H17ClN2OS |
| Molecular Weight | 332.85 |
| SMILES | ClC1=CC2=C(N=C3C=CC(OC)=CC3=C2SCCCN)C=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.