Fig. 1 · Structure
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Lobradimil
Bradykinin B2 Receptor Agonist
Lobradimil, a synthetic bradykinin analog, acts as a potent and selective agonist of the bradykinin B2 receptor (Ki: 0.54 nM). This compound enhances blood-brain barrier permeability, making it valuable for investigations into neuropharmacology and brain tumor research. Its unique properties facilitate studies aimed at drug delivery across the blood-brain barrier and potential therapeutic applications in CNS disorders.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 159768-75-9 |
| Applications | Bradykinin B2 Receptor Agonist |
| Formula | C49H75N15O12S |
| Molecular Weight | 1098.28 |
| Synonyms | RMP 7 |
| SMILES | COc1ccc(C[C@@H](CN[C@@H](CCCNC(N)=N)C(O)=O)NC(=O)[C@@H]2CCCN2C(=O)[C@H](CO)NC(=O)[C@H](Cc2cccs2)NC(=O)CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H]2CCCN2C(=O)[C@@H](N)CCCNC(N)=N)cc1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.