Documents & Downloads

LU-25-077

M1 Agonist

LU-25-077 is a brain-penetrant N-demethyl metabolite of Lu 25-109, functioning primarily as a partial agonist of the M1 muscarinic acetylcholine receptor while exhibiting antagonistic properties toward M2 and M3 receptors. This compound is valuable for neurological research, enabling the exploration of cholinergic modulation in various pathophysiological conditions. It provides an important tool for studying cognitive processes and potential therapeutic strategies for neurodegenerative disorders.

Out of Stock

Free Aliquoting for Your Order

Tell us your preferred amount per vial. We’ll confirm the options.

Specifications

Manufacturer	Adooq Bioscience
Actions	Partial Agonist
CAS Number	221549-70-8
Applications	M1 Agonist
Formula	C₈H₁₃N₅
Molecular Weight	179.22
SMILES	CCN1N=NC(C2=CCCNC2)=N1

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.