LY2157299

Catalog No.: A11017

TGF-βR Inhibitor

LY2157299 Chemical Structure

CAS NO. 700874-72-2

LY2157299 is an orally active transforming growth factor beta receptor (TGF-βR) kinase inhibitor.

Availability: In stock

Package Price Qty
5 mg
$45.00
10 mg
$65.00
25 mg
$140.00
100 mg
$260.00
10mM * 1mL in DMSO
$70.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

LY2157299 is an orally active transforming growth factor beta receptor (TGF-βR) kinase inhibitor.
Targets
TβRI (Cell-free assay)
56 nM
In vitro DMSO 74 mg/mL (200.31 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.07 mL 135.35 mL 270.71 mL
0.5 mM 5.41 mL 27.07 mL 54.14 mL
1 mM 2.71 mL 13.54 mL 27.07 mL
5 mM 0.54 mL 2.71 mL 5.41 mL

*The above data is based on the productmolecular weight 369.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11017
Actions Inhibitor
M. Wt 369.4
Formula C22H19N5O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 700874-72-2
Synonyms LY-2157299
SMILES CC1=CC=CC(=N1)C2=NN3CCCC3=C2C4=C5C=C(C=CC5=NC=C4)C(=O)N

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