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TGF-βR Inhibitor

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Catalog No. A11017

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
LY2157299 5mg A11017-5

Regular Price: $90.00

Special Price: $81.00

LY2157299 10mg A11017-10

Regular Price: $135.00

Special Price: $121.50

LY2157299 25mg A11017-25

Regular Price: $270.00

Special Price: $243.00

LY2157299 100mg A11017-100

Regular Price: $750.00

Special Price: $675.00

LY2157299 10mM * 1mL in DMSO A11017-10mM-D

Regular Price: $125.00

Special Price: $112.50

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

LY2157299 is an orally active transforming growth factor beta receptor (TGF-βR) kinase inhibitor.


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Publications citing Adooq Products
LY2157299 Citations (1)
  • Oguri G, .et al. Effects of methylglyoxal on human cardiac fibroblast: roles of transient receptor potential ankyrin 1 (TRPA1) channels., Am J Physiol Heart Circ Physiol., 2014, 307(9):H1339-52 PMID: 25172898

Chemical Information

Catalog Num A11017
Actions Inhibitor
M. Wt 369.4
Formula C22H19N5O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 700874-72-2
Synonyms LY-2157299

Biological Activity

LY2157299 is an orally active transforming growth factor beta receptor (TGF-βR) kinase inhibitor.
TβRI (Cell-free assay)
56 nM


Solubility (25°C)* In vitro DMSO 74 mg/mL (200.31 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.07 mL 135.35 mL 270.71mL
0.5 mM 5.41 mL 27.07 mL 54.14 mL
1 mM 2.71 mL 13.54 mL 27.07 mL
5 mM 0.54 mL 2.71 mL 5.41 mL

*The above data is based on the productmolecular weight 369.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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