Fig. 1 · Structure
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LY219057
CCK-8 Antagonist
LY219057 is a potent antagonist of cholecystokinin octapeptide (CCK-8), exhibiting an ID50 of 287.5 nM. This compound interferes with CCK-8 signaling pathways, making it valuable for investigating gastrointestinal and central nervous system functions. Its application spans research into appetite regulation, digestive processes, and potential therapeutic strategies for related disorders.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 150351-93-2 |
| Applications | CCK-8 Antagonist |
| Formula | C23H17ClF3N3OS |
| Molecular Weight | 475.91 |
| SMILES | FC(F)(F)C(C=C1NC(N2[C@@H](C3=CC=CC=C3)[C@H](C4=CC=CC=C4)C(N2)=O)=S)=C(C=C1)Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.