LY317615 (Enzastaurin)

Name: LY317615 (Enzastaurin)
SKU: A10356
Price: 30 USD
Rating: 5 (1 reviews)

Catalog No.: A10356

PKCβ inhibitor

Adooq's LY317615 (Enzastaurin) has been cited by 1 publications

LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).

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Grouped product items
Size	Price	Stock
5mg	$30.00	In stock
10mg	$40.00	In stock
25mg	$80.00	In stock
50mg	$115.00	In stock
100mg	$190.00	In stock
200mg	$345.00	In stock
*10mM 1mL in DMSO**	$40.00	In stock
Bulk Size	Bulk Discount

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Important Notice: For research use only. We do not sell to patients.

Data Sheet

SDS

Adooq Products cited in reputable paper

Adooq's LY317615 (Enzastaurin) has been cited by 1 publications

Bopei Cui, .et al. , Signal Transduct Target Ther, 2023, Sep 25;8(1):366 PMID: 37743418

Biological Activity

Discription

LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).

Targets

Target	Value

Product Information

Catalog Num	A10356
Formula	C32H29N5O2
Molecular Weight	515.6
CAS Number	170364-57-5
SMILES	CN1C=C(C2=CC=CC=C21)C3=C(C(=O)NC3=O)C4=CN(C5=CC=CC=C54)C6CCN(CC6)CC7=CC=CC=N7
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro (25°C)	DMSO	29 mg/mL (56.24 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	15% Captisol	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	19.39 mL	96.97 mL	193.95 mL
0.5 mM	3.88 mL	19.39 mL	38.79 mL
1 mM	1.94 mL	9.7 mL	19.39 mL
5 mM	0.39 mL	1.94 mL	3.88 mL

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