LY317615 (Enzastaurin)

Catalog No.: A10356

PKCβ inhibitor

LY317615 (Enzastaurin)

LY317615 (Enzastaurin) Chemical Structure

CAS NO. 170364-57-5

LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).

Availability: In stock

Package Price Qty
10 mg

Regular Price: $40.00

Special Price $32.00

50 mg

Regular Price: $120.00

Special Price $96.00

100 mg

Regular Price: $200.00

Special Price $160.00

200 mg

Regular Price: $350.00

Special Price $280.00

10mM * 1mL in DMSO
$80.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Details

LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).
Targets
PKCβ (Cell-free assay) PKCα (Cell-free assay) PKCγ (Cell-free assay) PKCε (Cell-free assay)
6 nM39 nM83 nM110 nM
In vitro (25°C) DMSO 30 mg/mL (58.18 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 15% Captisol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.39 mL 96.97 mL 193.95 mL
0.5 mM 3.88 mL 19.39 mL 38.79 mL
1 mM 1.94 mL 9.7 mL 19.39 mL
5 mM 0.39 mL 1.94 mL 3.88 mL

*The above data is based on the productmolecular weight 515.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

Catalog Num A10356
Actions Inhibitor
M. Wt 515.6
Formula C32H29N5O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 170364-57-5
Synonyms LY-317615
SMILES CN1C=C(C2=CC=CC=C21)C3=C(C(=O)NC3=O)C4=CN(C5=CC=CC=C54)C6CCN(CC6)CC7=CC=CC=N7

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