Fig. 1 · Structure
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M1 mAChR modulator-1
M1 mAChR Positive Allosteric Modulator
M1 mAChR modulator-1 is a positive allosteric modulator of the muscarinic M1 receptor (mAChR1). It enhances gastrointestinal motility and facilitates defecation in mouse models, exhibiting low permeability to the central nervous system. This compound is valuable for research focused on gastrointestinal disorders, particularly constipation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Modulator |
| CAS Number | 2247999-07-9 |
| Applications | M1 mAChR Positive Allosteric Modulator |
| Formula | C26H30FN3O5 |
| Molecular Weight | 483.53 |
| SMILES | O=C(C(C=CC(CC(C=C1C(N=CN(C1=O)[C@H]2CCOC[C@@H]2O)=C3C)=C3C)=C4)=C4F)NCCOC |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.