Fig. 1 · Structure
Documents & Downloads
M617
GAL1 Agonist
M617 is a selective galanin receptor 1 (GAL1) agonist, exhibiting inhibition constants (Kis) of 0.23 nM and 5.71 nM for GAL1 and GAL2, respectively. This compound primarily targets GAL1 to promote GLUT4 expression, significantly enhancing GLUT4 content in the cardiac muscle of type 2 diabetic rats. M617 is useful in research focused on metabolic disorders and the modulation of glucose homeostasis.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 860790-38-1 |
| Applications | GAL1 Agonist |
| Formula | C112H161N29O28 |
| Molecular Weight | 2361.65 |
| SMILES | C([C@@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(NCC(N[C@@H](CC1=CC=C(O)C=C1)C(N[C@H](C(N[C@H](C(NCC(=O)N2[C@H](C(N[C@H](C(=O)N3[C@H](C(=O)N4[C@H](C(NCC(N[C@@H](CC5=CC=CC=C5)C(N[C@H](C(=O)N6[C@H](C(N[C@@H](CC7=CC=CC=C7)C(N[C@@H](CCCNC(=N)N)C(N)=O)=O)=O)CCC6)CO)=O)=O)=O)CCC4)CCC3)CCC(N)=O)=O)CCC2)=O)CC(C)C)=O)CC(C)C)=O)=O)=O)C)=O)CO)=O)CC(N)=O)=O)CC(C)C)=O)[C@@H](C)O)=O)NC(CN)=O)C=8C=9C(NC8)=CC=CC9 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.