MEK162 (ARRY-438162, Binimetinib)

Catalog No.: A11493

MEK1/2 inhibitor

MEK162 (ARRY-438162, Binimetinib)

MEK162 (ARRY-438162, Binimetinib) Chemical Structure

CAS NO. 606143-89-9

MEK162 (ARRY-438162) is a potent, selective, ATP uncompetitive inhibitor of MEK1/2.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $40.00

Special Price $32.00

10 mg

Regular Price: $60.00

Special Price $48.00

25 mg

Regular Price: $100.00

Special Price $80.00

50 mg

Regular Price: $140.00

Special Price $112.00

10mM * 1mL in DMSO
$65.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Details

MEK162 (ARRY-438162) is a potent, selective, ATP uncompetitive inhibitor of MEK1/2.
Targets
MEK
12 nM
In vitro (25°C) DMSO 88 mg/mL (199.44 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 1% CMC/0.5% Tween-80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.73 mL 113.64 mL 227.27 mL
0.5 mM 4.55 mL 22.73 mL 45.45 mL
1 mM 2.27 mL 11.36 mL 22.73 mL
5 mM 0.45 mL 2.27 mL 4.55 mL

*The above data is based on the productmolecular weight 440.0 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

Catalog Num A11493
Actions Inhibitor
M. Wt 440.0
Formula C17H15BrF2N4O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 606143-89-9
Synonyms ARRY-162, MEK-162, MEK 162
SMILES CN1C=NC2=C1C=C(C(=C2F)NC3=C(C=C(C=C3)Br)F)C(=O)NOCCO

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