Fig. 1 · Structure
Documents & Downloads
MK-2295
Cat. No.
A68828
CAS
573678-04-3
TRPV1 Antagonist
MK-2295 (NGD-8243) is a potent TRPV1 antagonist that plays a crucial role in pain modulation. Its primary biological activity is as an analgesic agent, making it a valuable tool for research aimed at understanding and addressing pain mechanisms. MK-2295 is useful in studies exploring the therapeutic potential of TRPV1 inhibition in various pain-related conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 573678-04-3 |
| Applications | TRPV1 Antagonist |
| Formula | C21H12F6N4 |
| Molecular Weight | 434.34 |
| Synonyms | NGD-8243 |
| SMILES | C1=CC(=C(N=C1)C2=CC3=C(C=C2)C(=NC=N3)NC4=CC=C(C=C4)C(F)(F)F)C(F)(F)F |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.