MPEP

Catalog No.: A12589

mGlu5 receptor antagonist

MPEP

MPEP Chemical Structure

CAS NO. 96206-92-7

MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors.

Availability: In stock

Package Price Qty
10 mg

Regular Price: $50.00

Special Price $40.00

25 mg

Regular Price: $100.00

Special Price $80.00

50 mg

Regular Price: $160.00

Special Price $128.00

100 mg

Regular Price: $280.00

Special Price $224.00

10mM * 1mL in DMSO
$70.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Details

MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors.
Targets
mGluR5
36 nM
In vitro DMSO 39 mg/mL (201.82 mM)
Water <1 mg/mL (<1 mM)
Ethanol 39 mg/mL (201.82 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 51.75 mL 258.73 mL 517.47 mL
0.5 mM 10.35 mL 51.75 mL 103.49 mL
1 mM 5.17 mL 25.87 mL 51.75 mL
5 mM 1.03 mL 5.17 mL 10.35 mL

*The above data is based on the productmolecular weight 193.249. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

Catalog Num A12589
Actions Antagonist
M. Wt 193.249
Formula C14H11N
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 96206-92-7
Synonyms N/A
SMILES CC1=CC=CC(=N1)C#CC2=CC=CC=C2

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