MPEP
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
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Discription | MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors. | ||
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Targets |
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Catalog Num | A12589 |
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Formula | C14H11N |
Molecular Weight | 193.249 |
CAS Number | 96206-92-7 |
SMILES | CC1=CC=CC(=N1)C#CC2=CC=CC=C2 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 36 mg/mL (186.3 mM) | |
Water | Insoluble | ||
Ethanol | 36 mg/mL (186.3 mM) | ||
In vivo | 2% DMSO+30% PEG 300+5% Tween 80 | 9 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 51.75 mL | 258.73 mL | 517.47 mL |
0.5 mM | 10.35 mL | 51.75 mL | 103.49 mL |
1 mM | 5.17 mL | 25.87 mL | 51.75 mL |
5 mM | 1.03 mL | 5.17 mL | 10.35 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2