Olcegepant

Catalog No.: A11512

CGRP1 receptor

Olcegepant

Olcegepant Chemical Structure

CAS NO. 204697-65-4

Olcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP.

Availability: In stock

Package Price Qty
2 mg
$81.00
5 mg
$162.00
10 mg
$315.00
50 mg
$927.00
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Biological Activity

Olcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 11.5 mL 57.49 mL 114.99 mL
0.5 mM 2.3 mL 11.5 mL 23 mL
1 mM 1.15 mL 5.75 mL 11.5 mL
5 mM 0.23 mL 1.15 mL 2.3 mL

*The above data is based on the productmolecular weight 869.65. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11512
CAS No. 204697-65-4
Formula C38H47Br2N9O5
M. Wt 869.65
Solubility DMSO
Purity >98%
Synonyms BIBN-4096; BIBN 4096BS
SMILES O=C1N(CC2=C(N1)C=CC=C2)C3CCN(C(N[[email protected]@H](C(N[[email protected]](C(N4CCN(C5=CC=NC=C5)CC4)=O)CCCCN)=O)CC6=CC(Br)=C(C(Br)=C6)O)=O)CC3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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