ORM-15341

Catalog No.: A12312

human AR (hAR) antagonist

ORM-15341

ORM-15341 Chemical Structure

CAS NO. 1297537-33-7

ORM-15341 is a potent and full antagonist for human AR (hAR) with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells stably expressing full-length hAR and an androgen-responsive luciferase reporter gene construct.

Availability: In stock

Package Price Qty
5 mg
$315.00
10 mg
$543.00
50 mg
$1,610.00
100 mg
$3,220.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

ORM-15341 is a potent and full antagonist for human AR (hAR) with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells stably expressing full-length hAR and an androgen-responsive luciferase reporter gene construct.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.2 mL 126 mL 252 mL
0.5 mM 5.04 mL 25.2 mL 50.4 mL
1 mM 2.52 mL 12.6 mL 25.2 mL
5 mM 0.5 mL 2.52 mL 5.04 mL

*The above data is based on the productmolecular weight 396.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12312
Actions Antagonist
CAS No. 1297537-33-7
Formula C19H17ClN6O2
M. Wt 396.83
Purity >98%
Synonyms ORM15341, ORM 15341
SMILES ClC1=C(C#N)C=CC(C2=NN(C[[email protected]](C)NC(C3=NNC(C(C)=O)=C3)=O)C=C2)=C1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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