Other Inhibitors

Other Inhibitors groups bioactive small molecules whose targets fall outside the pathway categories of this catalogue. The compounds have not yet been assigned to target categories, so the range is broad and uneven. Streptozotocin, a glucosamine-nitrosourea compound used to induce experimental diabetes in rodents, sits beside the O-GlcNAcase inhibitor Thiamet G. Exherin is an N-cadherin antagonist, and AdipoRon is an agonist of adiponectin receptors 1 and 2 (AdipoR1 and AdipoR2). Plant compounds such as the isoflavone daidzein are also included. Despite the category name, not every compound is an inhibitor, as the AdipoRon example shows. Compounds with a well-defined target are usually listed in the matching pathway or target category.

5 Items

  • TOK-8801
    Cat. No.
    A12288

    TOK-8801

    TOK-8801 is a synthesized dihydroimidazothiazole carboxamide and is under development as an immunomodulator.

    1 mg
    $265.00
    5 mg
    $715.00
    All 6 sizes
  • Parimifasor
    Cat. No.
    A12594

    Parimifasor

    Synonyms: LYC30937

    Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.

    1 mg
    $35.00
    2 mg
    $50.00
    All 8 sizes
  • Plumbagin
    Cat. No.
    A15334

    Plumbagin

    Plumbagin, exhibits cytotoxicity in rodent models of carcinogenesis and carcinoma; has antifungal, antiviral, and antibacterial action.

    10 mg
    $25.00
    25 mg
    $45.00
    All 6 sizes
  • PZ-2891
    Cat. No.
    A18880

    PZ-2891

    PZ-2891 is an orally bioavailable, brain penetrant pantothenate kinase (PANK) modulator. PZ-2891 act as an orthosteric inhibitor at high concentrations and an allosteric activator at lower sub-saturating concentrations. PZ-2891 inhibits human pantothenate kinases PANK1β, PANK2, and PANK3 with IC50s of 40.2 nM, 0.7 nM and 1.3 nM, respectively.

    1 mg
    $25.00
    2 mg
    $40.00
    All 8 sizes
  • Velaresol
    Cat. No.
    A22668

    Velaresol

    Velaresol, also known as BW12C or BW12C79, is a oxyhaemoglobin stabilizer.

    5 mg
    $30.00
    10 mg
    $55.00
    All 6 sizes

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