Drug Derivative

Cat. No.

A25665

CAS No.

2699713-95-4

rel-Latanoprost acid

rel-Latanoprost acid is a relative configuration of Latanoprost acid. Latanoprost acid, an analog of prostaglandin (PG) F2α, is an selective prostanoid receptor (FP) agonist that specifically activates the FP-PG receptor. Latanoprost acid inhibits RANKL-induced osteoclastgenesis and function by inhibiting ERK, AKT, JNK, and p38 cascade, following by the c-fos/NFATc1 pathway. Latanoprost acid is a medication which works to lower pressure inside the eyes.

Cat. No.

A93198

CAS No.

61423-61-8

2-Aminoethyl ((R)-2,3-bis(hexadecyloxy)propyl) hydrogen phosphate

2-Aminoethyl ((R)-2,3-bis(hexadecyloxy)propyl) hydrogen phosphate functions as an ester product. This compound is utilized in biochemical research for its role in lipid-based systems and as a potential modulator of cellular membrane dynamics. Its application extends to studies on membrane biophysics and the design of novel drug delivery systems.

Cat. No.

A93454

CAS No.

3158-47-2

6-Hydroxyoctadecanoic acid

6-Hydroxyoctadecanoic acid is a fatty acid derivative characterized by its hydroxyl group at the sixth carbon position. This compound exhibits significant biological activity as a potential modulator of lipid metabolism and plays a role in cell signaling pathways. It is utilized in various research applications including studies on metabolic diseases, lipid biochemistry, and the development of novel therapeutic agents targeting metabolic disorders.

Cat. No.

A93483

CAS No.

911634-03-2

Methyl 14(S),15(S)-epoxy-11(R,S)-hydroxy-5(Z),8(Z),12(E)-eicosatrienoate

Methyl 14(S),15(S)-epoxy-11(R,S)-hydroxy-5(Z),8(Z),12(E)-eicosatrienoate is a bioactive ester compound. It serves as a significant modulator of lipid metabolism and is utilized in research focused on lipid signaling pathways. This compound may be applicable in studies exploring the roles of fatty acid derivatives in cellular processes and their implications in various diseases.

Cat. No.

A93713

CAS No.

2692623-71-3

Palmitoleyl arachidonate

Palmitoleyl arachidonate is an ester product primarily involved in lipid metabolism. This compound serves as a potential modulator of membrane fluidity and cell signaling pathways influenced by fatty acid composition. Its unique structural properties make it valuable for research into metabolic processes and cellular responses to various stimuli. Researchers may utilize palmitoleyl arachidonate in studies focusing on inflammation, cardiovascular health, and lipid-related disorders.

Cat. No.

A95447

CAS No.

105080-32-8

ICI 200355

ICI 200355 is a potent drug derivative that acts as a selective estrogen receptor modulator (SERM). It demonstrates significant biological activity in modulating estrogenic effects and is primarily utilized in research focused on hormone-related disorders and cancer therapy. This compound serves as an important tool in studying the mechanisms of estrogen receptor signaling and therapeutic approaches for estrogen-dependent tumors.

Cat. No.

A95457

CAS No.

155432-64-7

TAK 187

TAK 187 is a drug derivative that exhibits potent activity as a selective modulator in targeted therapeutic applications. This compound has been shown to influence key biological pathways, making it relevant for research focused on drug development and pathway elucidation in various disease models. Its unique mechanism of action offers promising insights for investigating therapeutic strategies in complex biological systems.

Cat. No.

A95460

CAS No.

62622-76-8

RU 25434

RU 25434 is a drug derivative that acts as a modulator of specific signaling pathways. This compound has demonstrated significant biological activity in various in vitro studies, making it a valuable tool for researchers investigating cellular responses related to drug mechanisms. RU 25434 is primarily utilized in pharmacological research to explore its therapeutic potential and effects on disease models.

Cat. No.

A95515

CAS No.

868273-09-0

Org 27759

Org 27759 is a potent drug derivative known for its role as a selective modulator. This compound exhibits significant biological activity, making it a valuable tool for investigating therapeutic mechanisms and pathways. It is widely utilized in drug discovery and development research, particularly in studies aimed at optimizing pharmacological profiles and enhancing drug efficacy.

Cat. No.

A95560

CAS No.

301648-08-8

Hydro-UCB35625

Hydro-UCB35625 is a drug derivative that primarily acts as a modulator of specific biological pathways. This compound exhibits notable activity in cellular assays and has potential applications in pharmacological research. Its unique mechanism makes it a valuable tool for studying drug interactions and therapeutic effects in various biological contexts.

Cat. No.

A95631

CAS No.

143782-25-6

RU 56187

RU 56187 is a drug derivative that acts as a selective modulator of cellular pathways. This compound exhibits significant biological activity, making it valuable for investigations into cellular signaling mechanisms. It is commonly utilized in research applications focused on pharmacology and drug development.

Cat. No.

A95641

CAS No.

2231302-46-6

5-HT4R agonist-1

5-HT4R agonist-1 is a selective agonist for the 5-hydroxytryptamine 4 receptor (5-HT4R), a target involved in various neuropharmacological processes. This compound exhibits significant biological activity in modulating gastrointestinal motility and cognitive functions. It serves as a valuable tool in research applications focused on gastrointestinal disorders and neurodegenerative diseases, aiding in the exploration of therapeutic strategies targeting the serotonergic system.

Cat. No.

A95721

CAS No.

127682-75-1

Ro24-5098

Ro24-5098 is a potent drug derivative that functions as a selective modulator of the sigma-1 receptor. This compound has demonstrated significant biological activity in various cellular models, providing insights into neuroprotective mechanisms and potential therapeutic applications for neurodegenerative diseases. Researchers may utilize Ro24-5098 to investigate pathways involving sigma-1 receptor signaling and its implications in drug development and disease treatment.

Cat. No.

A95844

CAS No.

105748-60-5

Methoxybrassinin

Synonyms: 1-Methoxybrassinin

Methoxybrassinin is a bioactive derivative of brassinosteroids that functions primarily as a modulator of plant growth and development. This compound exhibits key biological activities including promoting cell division and elongation, enhancing stress tolerance, and influencing gene expression in response to environmental stimuli. Research applications for Methoxybrassinin include studying its effects on plant physiology, exploring mechanisms of stress resistance, and investigating its potential in agricultural biotechnology.

Cat. No.

A96051

CAS No.

42863-81-0

Lopirazepam

Synonyms: D-12524

Lopirazepam is a benzodiazepine derivative that primarily acts as a positive allosteric modulator of GABA-A receptors. It exhibits anxiolytic and sedative properties, making it valuable for research into anxiety disorders and sleep regulation. This compound is useful for studying the pharmacological effects of benzodiazepines and their potential therapeutic applications in neuropharmacology.

Cat. No.

A96248

CAS No.

884599-96-6

γ-Secretase modulator 16

γ-Secretase modulator 16 is a selective modulator of the γ-secretase complex, primarily targeting the processing of amyloid precursor protein (APP). This compound is known to influence the production of amyloid-beta peptides, thereby playing a crucial role in the modulation of neurodegenerative pathways associated with Alzheimer's disease. It serves as a valuable tool for research aimed at understanding γ-secretase function and the development of therapeutic strategies for Alzheimer’s and other related disorders.

Cat. No.

A96256

CAS No.

937395-09-0

BX048

BX048 is a potent drug derivative that acts as a selective modulator of target pathways. This compound exhibits significant biological activity, making it suitable for various research applications, including pharmacological studies and mechanism of action investigations. Researchers can utilize BX048 to explore its effects on cellular processes and therapeutic potential in specific disease models.

Cat. No.

A96305

CAS No.

114800-19-0

WEB2347

WEB2347 is a drug derivative that functions primarily as a selective modulator of cellular signaling pathways. This compound exhibits significant biological activity in the regulation of immune responses and has potential applications in the study of inflammation and cancer therapeutics. Researchers use WEB2347 to explore its effects on various cellular processes and to develop novel treatments targeting specific pathways implicated in disease.

Cat. No.

A96372

CAS No.

2803608-05-9

STING agonist-49-CO-C2-mal-Cys

STING agonist-49-CO-C2-mal-Cys is a derivative of the STING agonist designed to facilitate the catabolism of antibody-drug conjugates (ADCs) and promote payload release. This compound exhibits significant antitumor activity in vivo, making it a valuable tool in cancer research. Its unique structure provides essential interactions with target proteins and E3 ligases, contributing to its efficacy in therapeutic applications.

Cat. No.

A96413

CAS No.

65934-61-4

RU 24926

RU 24926 is a drug derivative that functions primarily as a selective agonist for the corticotropin-releasing hormone receptor 1 (CRHR1). This compound exhibits key biological activity in modulating stress responses and has been utilized in research related to anxiety and depression models. RU 24926 serves as an important tool for investigating the pathways involved in neuroendocrine regulation and stress-related disorders.

Cat. No.

A96442

CAS No.

142023-57-2

BIBS-222

BIBS-222 is a drug derivative that acts as a potent modulator of various biological pathways. It exhibits significant pharmacological activity, making it a valuable tool for research into therapeutic mechanisms and drug development. BIBS-222 can be utilized in studies focusing on drug efficacy, target interactions, and the exploration of molecular targets in disease models.

Cat. No.

A96485

CAS No.

104493-13-2

Adecypenol

Synonyms: OM-3223

Adecypenol is a drug derivative that acts as a selective modulator of various biological pathways. It exhibits significant activity in altering drug metabolism and can be used in pharmacological research to investigate the impact of drug modifications on efficacy and toxicity. This compound is valuable for studies focusing on drug development and optimization.

Cat. No.

A96515

CAS No.

845555-94-4

MNI-D-aspartate

MNI-D-aspartate is a potent drug derivative that acts as an NMDA receptor agonist. It plays a critical role in neurotransmission and is vital for studies related to excitatory signaling in the central nervous system. Research applications include investigations into neuropharmacology and the modulation of synaptic plasticity, making it valuable for understanding various neurological conditions.

Cat. No.

A96523

CAS No.

90505-66-1

Ro 16-8714

Ro 16-8714 is a drug derivative that functions primarily as a selective modulator of various biological signaling pathways. This compound exhibits significant biological activity in cellular models, making it a valuable tool for investigating mechanism of action studies and drug discovery. Its ability to interact with specific targets allows for exploration of therapeutic strategies in diverse research applications.

Cat. No.

A96857

CAS No.

88594-08-5

CD-349

CD-349 is a potent drug derivative that functions primarily as a modulator of key biological pathways. It exhibits significant biological activity, making it suitable for various research applications, including drug discovery and development. Researchers may utilize CD-349 to explore its effects on cellular mechanisms and pharmacological properties, providing valuable insights into its therapeutic potential.