Drug Derivative

Cat. No.

A25665

CAS No.

2699713-95-4

rel-Latanoprost acid

rel-Latanoprost acid is a relative configuration of Latanoprost acid. Latanoprost acid, an analog of prostaglandin (PG) F2α, is an selective prostanoid receptor (FP) agonist that specifically activates the FP-PG receptor. Latanoprost acid inhibits RANKL-induced osteoclastgenesis and function by inhibiting ERK, AKT, JNK, and p38 cascade, following by the c-fos/NFATc1 pathway. Latanoprost acid is a medication which works to lower pressure inside the eyes.

Cat. No.

A67079

CAS No.

150465-29-5

L-Cysteine S-sulfate sodium hydrate

L-Cysteine S-sulfate sodium hydrate is an S-sulfated derivative of L-cysteine and serves as a substrate for cystine lyase. This compound is utilized in mass spectrometry and chromatography analyses, making it valuable for biochemical research. Its unique structure allows for the investigation of cysteine metabolism and related pathways in cellular biology.

Cat. No.

A89500

CAS No.

108045-15-4

Heptaprenyl-MPDA

Synonyms: Heptaprenyl phosphate

Heptaprenyl-MPDA is an ester product that acts as an endogenous substrate for Phospho-MurNAc-pentapeptide translocase (MraY). This compound plays a critical role in bacterial cell wall biosynthesis and is valuable for research into bacterial infections. Its unique structure and function make it an essential tool for studies aimed at understanding antimicrobial mechanisms and developing new therapeutic strategies.

Cat. No.

A93338

CAS No.

111278-02-5

Hexadecanedioyl-mono-coenzyme A

Hexadecanedioyl-mono-coenzyme A is an ester product that serves as a substrate in fatty acid metabolism. This compound is involved in the synthesis and degradation of lipids, making it essential for research in metabolic pathways and energy storage mechanisms. Its role in enzymatic reactions can be leveraged in studies focusing on lipid biology and related metabolic disorders.

Cat. No.

A94240

CAS No.

162040-64-4

Valeryl-L-carnitine chloride

Valeryl-L-carnitine chloride is an ester derivative of L-carnitine, primarily functioning as a carnitine acyltransferase substrate. Its biological activity includes the facilitation of fatty acid transport into mitochondria, playing a crucial role in energy metabolism. This compound is utilized in research focused on metabolic disorders, mitochondrial dysfunction, and the study of fatty acid oxidation.

Cat. No.

A95641

CAS No.

2231302-46-6

5-HT4R agonist-1

5-HT4R agonist-1 is a selective agonist for the 5-hydroxytryptamine 4 receptor (5-HT4R), a target involved in various neuropharmacological processes. This compound exhibits significant biological activity in modulating gastrointestinal motility and cognitive functions. It serves as a valuable tool in research applications focused on gastrointestinal disorders and neurodegenerative diseases, aiding in the exploration of therapeutic strategies targeting the serotonergic system.

Cat. No.

A96372

CAS No.

2803608-05-9

STING agonist-49-CO-C2-mal-Cys

STING agonist-49-CO-C2-mal-Cys is a derivative of the STING agonist designed to facilitate the catabolism of antibody-drug conjugates (ADCs) and promote payload release. This compound exhibits significant antitumor activity in vivo, making it a valuable tool in cancer research. Its unique structure provides essential interactions with target proteins and E3 ligases, contributing to its efficacy in therapeutic applications.

Cat. No.

A96413

CAS No.

65934-61-4

RU 24926

RU 24926 is a drug derivative that functions primarily as a selective agonist for the corticotropin-releasing hormone receptor 1 (CRHR1). This compound exhibits key biological activity in modulating stress responses and has been utilized in research related to anxiety and depression models. RU 24926 serves as an important tool for investigating the pathways involved in neuroendocrine regulation and stress-related disorders.

Cat. No.

A96515

CAS No.

845555-94-4

MNI-D-aspartate

MNI-D-aspartate is a potent drug derivative that acts as an NMDA receptor agonist. It plays a critical role in neurotransmission and is vital for studies related to excitatory signaling in the central nervous system. Research applications include investigations into neuropharmacology and the modulation of synaptic plasticity, making it valuable for understanding various neurological conditions.

Cat. No.

A97088

CAS No.

98537-38-3

β-Methoxy 2C-D hydrochloride

β-Methoxy 2C-D hydrochloride is a phenethylamine derivative that functions primarily as a selective serotonin receptor agonist. This compound exhibits psychoactive properties and has potential applications in neuroscience research, particularly in the study of serotonin modulation and its effects on behavior. β-Methoxy 2C-D hydrochloride serves as a valuable tool for investigating the pharmacological profiles of serotonin receptor activity and related signaling pathways.

Cat. No.

B18253

CAS No.

17363-90-5

Para-nitrophenyl oleate

Para-nitrophenyl oleate is an ester compound known for its role as a substrate in enzymatic assays. It acts as a colorimetric indicator for lipases, facilitating the measurement of their activity in biochemical research. This reagent is widely utilized in studies involving lipid metabolism and enzyme kinetics.