Fig. 1 · Structure
Documents & Downloads
PCAF-IN-2
PCAF Inhibitor
PCAF-IN-2 is a potent inhibitor of PCAF (p300/CBP-associated factor) with an IC50 value of 5.31 µM. This compound demonstrates significant anti-tumor activity, inducing apoptosis and effectively arresting the cell cycle at the G2/M phase. PCAF-IN-2 is valuable for research applications focused on cancer biology and the modulation of gene expression pathways.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 56173-05-8 |
| Applications | PCAF Inhibitor |
| Formula | C10H7F3N6 |
| Molecular Weight | 268.20 |
| SMILES | FC(C1=NN=C2N1N=C(NN)C3=C2C=CC=C3)(F)F |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.