Fig. 1 · Structure
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Pentoxyverine citrate
Sigma-1 Receptor Agonist
Pentoxyverine citrate is a sigma-1 receptor agonist that effectively crosses the blood-brain barrier. With binding affinities of 41 nM for σ1, it demonstrates potent antitussive, anticonvulsant, and spasmolytic activities. This compound is utilized in research for its ability to inhibit bronchial interceptor activity, attenuate cough reflex, relax bronchial smooth muscle, and reduce airway resistance, making it valuable in the study of respiratory conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 23142-01-0 |
| Applications | Sigma-1 Receptor Agonist |
| Formula | C26H39NO10 |
| Molecular Weight | 525.59 |
| Synonyms | Carbetapentane citrate |
| SMILES | O=C(C1(C2=CC=CC=C2)CCCC1)OCCOCCN(CC)CC.O=C(CC(C(O)=O)(O)CC(O)=O)O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.