Fig. 1 · Structure
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PGN-9856
EP2 receptor Agonist
PGN-9856 is a selective agonist of the EP2 receptor, exhibiting high affinity with a pKi of 8.3 or greater. This potent non-prostanoid compound demonstrates significant biological activity, with an EC50 value of 8.5 or higher, making it effective in anti-inflammatory and anti-glaucoma research applications. PGN-9856 serves as a valuable tool for exploring the therapeutic potential of targeting the EP2 receptor in various pharmacological studies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 863704-91-0 |
| Applications | EP2 receptor Agonist |
| Formula | C21H15F2NO4 |
| Molecular Weight | 383.34 |
| SMILES | O=C(O)COC1=CC=CC(NC(C2=CC(C3=CC=CC(F)=C3)=CC=C2F)=O)=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.