PI-103 Hydrochloride

Catalog No.: A15212

PI3K Inhibitor

PI-103 Hydrochloride

PI-103 Hydrochloride Chemical Structure

CAS NO. 371935-79-4

PI103 is a potent inhibitor with low IC50 values against recombinant PI3K isoforms p110alpha (IC50= 2 nM), p110beta (IC50= 3 nM), p110delta (IC50= 3 nM), and p110gamma (IC50= 15 nM), less potent to mTOR/DNA-PK with IC50 of 30 nM/23 nM.

Availability: In stock

Package Price Qty
10 mg
$65.00
50 mg
$200.00
100 mg
$360.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

PI103 is a potent inhibitor with low IC50 values against recombinant PI3K isoforms p110alpha (IC50= 2 nM), p110beta (IC50= 3 nM), p110delta (IC50= 3 nM), and p110gamma (IC50= 15 nM), less potent to mTOR/DNA-PK with IC50 of 30 nM/23 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.99 mL 129.93 mL 259.86 mL
0.5 mM 5.2 mL 25.99 mL 51.97 mL
1 mM 2.6 mL 12.99 mL 25.99 mL
5 mM 0.52 mL 2.6 mL 5.2 mL

*The above data is based on the productmolecular weight 384.82. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A15212
Actions Inhibitor
M. Wt 384.82
Formula C19H17ClN4O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 371935-79-4
Synonyms PI 103 hydrochloride, PI103 hydrochloride
SMILES C1COCCN1C2=NC(=NC3=C2OC4=C3C=CC=N4)C5=CC(=CC=C5)O.Cl

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