PI3Kδ/BET-IN-1

Name: PI3Kδ/BET-IN-1
Brand: Adooq Bioscience
SKU: A40402
Rating: 5 (288 reviews)

Catalog No.: A40402

PI3Kδ/BET Inhibitor

PI3Kδ/BET-IN-1 is a selective inhibitor targeting both PI3Kδ and the bromodomain BRD4-BD1. With an IC50 of 112 nM for PI3Kδ and 19 nM for BRD4-BD1, this compound demonstrates potent antiproliferative effects in diffuse large B-cell lymphoma (DLBCL) cells. Its dual inhibition mechanism makes it a valuable tool for research into cancer biology and therapeutic development.

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PI3Kδ/BET-IN-1 3054869-10-9 PI3Kδ/BET Inhibitor

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Biological Activity

Description	PI3Kδ/BET-IN-1 is a selective inhibitor targeting both PI3Kδ and the bromodomain BRD4-BD1. With an IC50 of 112 nM for PI3Kδ and 19 nM for BRD4-BD1, this compound demonstrates potent antiproliferative effects in diffuse large B-cell lymphoma (DLBCL) cells. Its dual inhibition mechanism makes it a valuable tool for research into cancer biology and therapeutic development.

Product Information

Catalog Num	A40402
Formula	C27H34N6O3S
Molecular Weight	522.66
CAS Number	3054869-10-9
SMILES	CN1C=C(C2=NC(N3CCOCC3)=C4SC(CN5CCC(C(C)(O)C)CC5)=CC4=N2)C6=C(C1=O)NC=C6

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