Pictilisib dimethanesulfonate

Catalog No.: A11444

PI3Kα/δ inhibitor

Pictilisib dimethanesulfonate

Pictilisib dimethanesulfonate Chemical Structure

CAS NO. 957054-33-0

Pictilisib dimethanesulfonate (GDC-0941 dimethanesulfonate) is a potent inhibitor of PI3Kα/δ with IC50 of 3 nM, with modest selectivity against p110β (11-fold) and p110γ (25-fold).

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50 mg
$81.00
100 mg
$140.00
500 mg
$414.00
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Biological Activity

Pictilisib dimethanesulfonate (GDC-0941 dimethanesulfonate) is a potent inhibitor of PI3Kα/δ with IC50 of 3 nM, with modest selectivity against p110β (11-fold) and p110γ (25-fold).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 14.17 mL 70.84 mL 141.67 mL
0.5 mM 2.83 mL 14.17 mL 28.33 mL
1 mM 1.42 mL 7.08 mL 14.17 mL
5 mM 0.28 mL 1.42 mL 2.83 mL

*The above data is based on the productmolecular weight 705.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11444
Actions Inhibitor
M. Wt 705.85
Formula C25H35N7O9S4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 957054-33-0
Synonyms GDC-0941 dimethanesulfonate; GDC-0941 2 MeSO3H salt
SMILES O=S(N1CCN(CC1)CC2=CC3=C(S2)C(N4CCOCC4)=NC(C5=CC=CC6=C5C=NN6)=N3)(C)=O.O=S(O)(C)=O.O=S(O)(C)=O

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