Fig. 1 · Structure
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Pristimerin
MGL Inhibitor
Pristimerin is a potent and reversible inhibitor of monoacylglycerol lipase (MGL), exhibiting an IC50 value of 93 nM. Its inhibition of MGL activity has been linked to potential therapeutic effects in pain management and inflammation. Pristimerin is valuable for research applications focused on the endocannabinoid system and lipid metabolism.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1258-84-0 |
| Applications | MGL Inhibitor |
| Formula | C30H40O4 |
| Molecular Weight | 464.64 |
| Synonyms | Celastrol methyl ester |
| SMILES | C[C@](C1=CC=C(C(C)=C2O)C3=CC2=O)(CC[C@]4(C)[C@@]5([H])C[C@@](C(OC)=O)(C)CC4)[C@]5(CC[C@]13C)C |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.