Fig. 1 · Structure
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PTAC oxalate
Muscarinic Receptor Ligand
PTAC oxalate is a selective ligand for muscarinic receptors, functioning as a partial agonist at M2 and M4 receptors while acting as an antagonist at M1, M3, and M5 receptors, with Ki values ranging from 0.2 to 2.8 nM in CHO cells. This compound demonstrates significant biological activity by alleviating mechanical allodynia associated with neuropathic pain and exhibiting potential antidepressant effects. PTAC oxalate serves as a valuable tool for research into muscarinic receptor function and the development of therapeutics for pain and mood disorders.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Partial Agonist |
| CAS Number | 201939-40-4 |
| Applications | Muscarinic Receptor Ligand |
| Formula | C14H21N3O4S2 |
| Molecular Weight | 359.46 |
| SMILES | CCCSC1=NSN=C1[C@@H]2[C@@H]3C[N@@](CCC3)C2.OC(C(O)=O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.