(R)-Elagolix

Catalog No.: A21184

GnRHR antagonist

(R)-Elagolix

(R)-Elagolix Chemical Structure

CAS NO. 834153-87-6

Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM).

Availability: In stock

Package Price Qty
2 mg

Regular Price: $54.00

Special Price $43.20

5 mg

Regular Price: $108.00

Special Price $86.40

10 mg

Regular Price: $210.00

Special Price $168.00

50 mg

Regular Price: $618.00

Special Price $494.40

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Biological Activity

Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 15.83 mL 79.17 mL 158.33 mL
0.5 mM 3.17 mL 15.83 mL 31.67 mL
1 mM 1.58 mL 7.92 mL 15.83 mL
5 mM 0.32 mL 1.58 mL 3.17 mL

*The above data is based on the productmolecular weight 631.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21184
Actions Antagonist
CAS No. 834153-87-6
Formula C32H30F5N3O5
M. Wt 631.59
Purity >98%
Synonyms NBI-56418, NBI56418, NBI 56418
SMILES FC1=C(C2=C(C)N(CC3=C(C(F)(F)F)C=CC=C3F)C(N(C[[email protected]](C4=CC=CC=C4)([H])NCCCC(O)=O)C2=O)=O)C=CC=C1OC
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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