(R,R,S)-GAT107 is a potent positive allosteric modulator of the α7 nicotinic receptors, exhibiting robust agonistic activity. This compound primarily functions through its (+)-isomer, demonstrating significant biological effects, while the (-)-isomer shows no such activity. Research indicates that (R,R,S)-GAT107 is currently recognized as the most effective ago-PAM for α7 nicotinic receptors, suggesting promising avenues for further investigation in vivo. Potential applications include studies related to cognitive enhancement and neuroinflammation.
(R,R,S)-GAT107 is a potent positive allosteric modulator of the α7 nicotinic receptors, exhibiting robust agonistic activity. This compound primarily functions through its (+)-isomer, demonstrating significant biological effects, while the (-)-isomer shows no such activity. Research indicates that (R,R,S)-GAT107 is currently recognized as the most effective ago-PAM for α7 nicotinic receptors, suggesting promising avenues for further investigation in vivo. Potential applications include studies related to cognitive enhancement and neuroinflammation.
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