Fig. 1 · Structure
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(Rac)-AMG 628
Cat. No.
A68870
CAS
862269-73-6
TRPV1 Antagonist
(Rac)-AMG 628 is a potent TRPV1 antagonist, exhibiting an IC50 of 3.7 nM. This compound is valuable for research in chronic pain mechanisms, providing insights into the role of TRPV1 in nociception and pain modulation. Its efficacy makes it a noteworthy tool for exploring potential therapeutic avenues in pain management.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 862269-73-6 |
| Applications | TRPV1 Antagonist |
| Formula | C25H25FN6O2S |
| Molecular Weight | 492.57 |
| SMILES | CC(NC1=NC2=C(OC3=NC=NC(N4CCN(C(C5=CC=C(F)C=C5)C)CC4)=C3)C=CC=C2S1)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.