(rac)-CHEMBL333994

Catalog No.: A59710
CCK-A Receptor Antagonist
(rac)-CHEMBL333994 is a potent Cholecystokinin A (CCK-A) receptor antagonist with an IC50 of 0.67 nM, demonstrating effective oral bioavailability. This compound selectively targets peripheral CCK receptors, making it valuable for studying mechanistic pathways involved in gastrointestinal disorders. Its ability to increase CCK mRNA levels positions (rac)-CHEMBL333994 as a useful tool in research aimed at understanding chronic pancreatitis and related conditions.
Grouped product items
Size Price Stock Qty
1mg
$155.00
In stock
2mg
$235.00
In stock
5mg
$395.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
Description(rac)-CHEMBL333994 is a potent Cholecystokinin A (CCK-A) receptor antagonist with an IC50 of 0.67 nM, demonstrating effective oral bioavailability. This compound selectively targets peripheral CCK receptors, making it valuable for studying mechanistic pathways involved in gastrointestinal disorders. Its ability to increase CCK mRNA levels positions (rac)-CHEMBL333994 as a useful tool in research aimed at understanding chronic pancreatitis and related conditions.
Product Information
Catalog NumA59710
FormulaC26H19FN4O2
Molecular Weight438.45
CAS Number126149-42-6
SMILESO=C(C(N1)=CC2=C1C=CC=C2)NC3C(N4C5=C(CC4)C=CC=C5C(C6=CC=CC=C6F)=N3)=O
Synonyms(rac)-FK-480
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