Regorafenib monohydrate

Catalog No.: A15218

Tyrosine kinase inhibitor

Regorafenib monohydrate

Regorafenib monohydrate Chemical Structure

CAS NO. 1019206-88-2

Regorafenib is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 of 13 nM/4.2 nM/46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM, respectively.

Availability: In stock

Package Price Qty
50 mg
$90.00
100 mg
$120.00
200 mg
$190.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Regorafenib is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 of 13 nM/4.2 nM/46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.97 mL 99.83 mL 199.67 mL
0.5 mM 3.99 mL 19.97 mL 39.93 mL
1 mM 2 mL 9.98 mL 19.97 mL
5 mM 0.4 mL 2 mL 3.99 mL

*The above data is based on the productmolecular weight 500.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A15218
Actions Inhibitor
M. Wt 500.83
Formula C21H17ClF4N4O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1019206-88-2
Synonyms BAY 73-4506 monohydrate
SMILES CNC(=O)C1=NC=CC(=C1)OC2=CC(=C(C=C2)NC(=O)NC3=CC(=C(C=C3)Cl)C(F)(F)F)F.O

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