Risotilide is a potent neprilysin inhibitor that effectively impedes enkephalinase B activity, with an IC50 value of 0.35 µM. Additionally, it demonstrates strong inhibition of enkephalinase A (IC50 = 0.02 µM) and aminopeptidase activity (IC50 = 13 µM). This comprehensive inhibition profile makes Risotilide a valuable reagent for studying enkephalin biodegradation and its implications in neurobiology and pain management research.
Risotilide is a potent neprilysin inhibitor that effectively impedes enkephalinase B activity, with an IC50 value of 0.35 µM. Additionally, it demonstrates strong inhibition of enkephalinase A (IC50 = 0.02 µM) and aminopeptidase activity (IC50 = 13 µM). This comprehensive inhibition profile makes Risotilide a valuable reagent for studying enkephalin biodegradation and its implications in neurobiology and pain management research.
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