Fig. 1 · Structure
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TEAD-IN-2
TEAD Inhibitor
TEAD-IN-2 is a selective inhibitor of the transcriptional enhancer associate domain (TEAD), functioning primarily through modulation via ubiquitination and degradation. This compound demonstrates significant biological activity in the regulation of TEAD-related pathways, making it a valuable tool for investigating various diseases and disorders linked to TEAD dysregulation. Its oral bioavailability allows for versatile application in preclinical studies aimed at understanding TEAD's role in cellular processes.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2563849-97-6 |
| Applications | TEAD Inhibitor |
| Formula | C16H18BrF3N2O |
| Molecular Weight | 391.23 |
| SMILES | FC(C1=CC=C(CN2CCC(C3CC(Br)=NO3)CC2)C=C1)(F)F |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.