Fig. 1 · Structure
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Telmapitant
NK1R Antagonist
Telmapitant is an orally active antagonist of the neurokinin-1 receptor (NK1R). This compound exhibits antiemetic properties, making it valuable for studying delayed onset emesis. It is utilized in research to investigate the mechanisms and treatment options related to nausea and vomiting.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 552292-58-7 |
| Applications | NK1R Antagonist |
| Formula | C24H23F6N3O3 |
| Molecular Weight | 515.45 |
| SMILES | O=C(N1)N[C@]2(CN[C@@](C3=CC=CC=C3)(CO[C@@H](C4=CC(C(F)(F)F)=CC(C(F)(F)F)=C4)C)CC2)C1=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.