Fig. 1 · Structure
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TG-2-IN-4
TG-2 Inhibitor
TG-2-IN-4 is a potent transglutaminase 2 (TG2) inhibitor, exhibiting an IC50 of less than 0.5 mM. This compound is suitable for investigating the role of TG2 in inflammatory disorders, facilitating research into potential therapeutic interventions and the underlying mechanisms of related diseases. TG-2-IN-4 serves as a valuable tool for studying the implications of TG2 activity in various biological contexts.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2410899-01-1 |
| Applications | TG-2 Inhibitor |
| Formula | C34H40N6O5 |
| Molecular Weight | 612.72 |
| SMILES | CC(C)CC1=C2C(N=C(N2)CN3C(C(NC([C@H](CC/C=C/C(N(C)C)=O)NC(OCC4=CC=CC=C4)=O)=O)=CC=C3)=O)=CC=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.