Fig. 1 · Structure
Documents & Downloads
TG2 inhibitor VA4
TG2 Inhibitor
TG2 inhibitor VA4 is an irreversible inhibitor of Type 2 transglutaminase (TG2). This compound selectively targets the transamidase site of TG2, effectively inhibiting both its transamidase and GTP-binding activities. TG2 inhibitor VA4 is utilized in research applications focused on fibrosis, neurodegenerative diseases, and cancer, facilitating the study of TG2's role in various biological processes.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2088001-23-2 |
| Applications | TG2 Inhibitor |
| Formula | C33H41N5O6S |
| Molecular Weight | 635.77 |
| SMILES | O=C(OCC1=CC=CC=C1)N[C@H](C(N2CCN(S(=O)(C3=C4C=CC=C(N(C)C)C4=CC=C3)=O)CC2)=O)CCCCNC(C=C)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.