TGR-1202 hydrochloride (Umbralisib HCl)

Name: TGR-1202 hydrochloride (Umbralisib HCl)
Brand: Adooq Bioscience
SKU: A16278
Rating: 5 (288 reviews)

Catalog No.: A16278

PI3Kδ inhibitor

TGR-1202 hydrochloride is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.

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TGR-1202 hydrochloride (Umbralisib HCl) 1532533-78-0 PI3Kδ inhibitor

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Grouped product items
Size	Price	Stock
2mg	$45.00	In stock
5mg	$100.00	In stock
10mg	$190.00	In stock
25mg	$400.00	In stock
50mg	$575.00	In stock
100mg	$980.00	In stock
Bulk Size	Bulk Discount

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Data Sheet SDS

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Biological Activity

Description

TGR-1202 hydrochloride is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.

Targets

Target	Value

Product Information

Catalog Num	A16278
Formula	C31H25ClF3N5O3
Molecular Weight	608.01
CAS Number	1532533-78-0
SMILES	O=C1C(C2=CC=CC(F)=C2)=C([C@@H](N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)C)OC6=CC=C(F)C=C16.[H]Cl
Synonyms	RP5264 hydrochloride, TGR1202 hydrochloride, TGR 1202 hydrochloride, RP-5264 hydrochloride, RP 5264 hydrochloride
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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