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TGR-1202 hydrochloride

PI3Kδ inhibitor

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Catalog No. A16278

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
TGR-1202 hydrochloride 5mg A16278-5
$120.00
TGR-1202 hydrochloride 10mg A16278-10
$220.00
TGR-1202 hydrochloride 50mg A16278-50
$580.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

TGR-1202 hydrochloride is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.

TGR-1202 hydrochloride

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Chemical Information

Catalog Num A16278
Actions Inhibitor
M. Wt 608.01
Formula C31H25ClF3N5O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1532533-78-0
Synonyms RP5264 hydrochloride, TGR1202 hydrochloride, TGR 1202 hydrochloride, RP-5264 hydrochloride, RP 5264 hydrochloride
SMILES O=C1C(C2=CC=CC(F)=C2)=C([[email protected]@H](N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)C)OC6=CC=C(F)C=C16.[H]Cl

Biological Activity

Description
TGR-1202 hydrochloride is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.45 mL 82.24 mL 164.47mL
0.5 mM 3.29 mL 16.45 mL 32.89 mL
1 mM 1.64 mL 8.22 mL 16.45 mL
5 mM 0.33 mL 1.64 mL 3.29 mL

*The above data is based on the productmolecular weight 608.01. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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