TGR-1202 (Umbralisib)

Catalog No.: A16277

PI3Kδ inhibitor

TGR-1202 (Umbralisib)

TGR-1202 (Umbralisib) Chemical Structure

CAS NO. 1532533-67-7

TGR-1202 is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.

Availability: In stock

Package Price Qty
5 mg
$120.00
10 mg
$220.00
50 mg
$580.00
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Biological Activity

TGR-1202 is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.5 mL 87.48 mL 174.96 mL
0.5 mM 3.5 mL 17.5 mL 34.99 mL
1 mM 1.75 mL 8.75 mL 17.5 mL
5 mM 0.35 mL 1.75 mL 3.5 mL

*The above data is based on the productmolecular weight 571.55. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16277
Actions Inhibitor
M. Wt 571.55
Formula C31H24F3N5O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1532533-67-7
Synonyms RP5264, TGR1202, TGR 1202, RP-5264, RP 5264
SMILES CC(C)OC1=C(C=C(C=C1)C2=NN(C3=C2C(=NC=N3)N)C(C)C4=C(C(=O)C5=C(O4)C=CC(=C5)F)C6=CC(=CC=C6)F)F

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