TPOP146

Catalog No.: A12655

CBP/P300 benzoxazepine bromodomain inhibitor

TPOP146

TPOP146 Chemical Structure

CAS NO. 2018300-62-2

TPOP146 is a selective CBP/P300 benzoxazepine bromodomain inhibitor with Kd values of 134 nM and 5.02 μM for CBP and BRD4.

Availability: In stock

Package Price Qty
5 mg
$95.00
10 mg
$163.00
50 mg
$483.00
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Biological Activity

TPOP146 is a selective CBP/P300 benzoxazepine bromodomain inhibitor with Kd values of 134 nM and 5.02 μM for CBP and BRD4.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.76 mL 103.82 mL 207.65 mL
0.5 mM 4.15 mL 20.76 mL 41.53 mL
1 mM 2.08 mL 10.38 mL 20.76 mL
5 mM 0.42 mL 2.08 mL 4.15 mL

*The above data is based on the productmolecular weight 481.58. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12655
Actions Inhibitor
CAS No. 2018300-62-2
Formula C27H35N3O5
M. Wt 481.58
Purity >98%
Synonyms TPOP-146; TPOP 146
SMILES COC1=CC(OC)=CC(C2=CC(C(N[[email protected]]3CCCN(C)C3)=O)=C(OCCN(C(CC)=O)C4)C4=C2)=C1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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