Fig. 1 · Structure
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TRPM8 antagonist 3
Cat. No.
A68758
CAS
2102179-29-1
TRP Channel Antagonist
TRPM8 Antagonist 3 is a selective antagonist targeting the Transient Receptor Potential Melastatin 8 (TRPM8) channel, exhibiting an IC50 value of 11 nM. This compound effectively inhibits TRPM8-mediated calcium influx, making it useful for studying nociceptive pathways and cold sensitivity. It has potential applications in research related to pain management, sensory biology, and neurobiology.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 2102179-29-1 |
| Applications | TRP Channel Antagonist |
| Formula | C13H12N2O4S |
| Molecular Weight | 292.31 |
| SMILES | O=C(N1OCCC1)C2=C(O)N=C(C3=C(O)C=CC=C3)S2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.