Fig. 1 · Structure
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TRPV4 antagonist 3
Cat. No.
A68824
CAS
2681273-35-6
TRPV4 Antagonist
TRPV4 antagonist 3 is a selective antagonist of the TRPV4 ion channel, demonstrating a pIC50 value of 8.4. This compound effectively inhibits TRPV4-mediated calcium influx, making it a valuable tool for investigating the physiological roles of TRPV4 in various biological processes. It has potential applications in pain research, inflammation studies, and the exploration of therapeutic strategies for TRPV4-related disorders.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 2681273-35-6 |
| Applications | TRPV4 Antagonist |
| Formula | C20H18F4N4O3S |
| Molecular Weight | 470.44 |
| SMILES | O=S(C1=CC=C(C#N)C=C1C(F)(F)F)(NCC[C@](C)(N)COC2=CC=C(C#N)C(F)=C2)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.