URAT1 inhibitor 2 is a potent inhibitor of the URAT1 transporter, exhibiting an IC50 of 1.36 µM for URAT1-mediated 14C-UA uptake, alongside effective inhibition of CYP1A2 and CYP2C9 with IC50 values of 16.97 µM and 5.22 µM, respectively. This compound demonstrates significant potential in the investigation of hyperuricemia and gout, making it a valuable tool for biochemical research and therapeutic development.
URAT1 inhibitor 2 is a potent inhibitor of the URAT1 transporter, exhibiting an IC50 of 1.36 µM for URAT1-mediated 14C-UA uptake, alongside effective inhibition of CYP1A2 and CYP2C9 with IC50 values of 16.97 µM and 5.22 µM, respectively. This compound demonstrates significant potential in the investigation of hyperuricemia and gout, making it a valuable tool for biochemical research and therapeutic development.
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