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Vapreotide acetate

Catalog No.: A61994
Neurokinin Receptor Antagonist
Vapreotide acetate is a neurokinin-1 (NK1) receptor antagonist, exhibiting an IC50 of 330 nM. This compound has demonstrated significant biological activity, making it valuable in the research of neurokinin signaling pathways and their roles in various physiological and pathological processes. Vapreotide acetate is commonly utilized in studies involving pain management, cancer therapy, and gastrointestinal disorders.
Vapreotide acetate 849479-74-9 Neurokinin Receptor Antagonist
Grouped product items
Size Price Stock Qty
1mg
$25.00
In stock
5mg
$50.00
In stock
10mg
$90.00
In stock
25mg
$165.00
In stock
50mg
$270.00
In stock
100mg
$425.00
In stock
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Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionVapreotide acetate is a neurokinin-1 (NK1) receptor antagonist, exhibiting an IC50 of 330 nM. This compound has demonstrated significant biological activity, making it valuable in the research of neurokinin signaling pathways and their roles in various physiological and pathological processes. Vapreotide acetate is commonly utilized in studies involving pain management, cancer therapy, and gastrointestinal disorders.
Product Information
Catalog NumA61994
FormulaC59H74N12O11S2
Molecular Weight1191.42
CAS Number849479-74-9
Sequence{d-Phe}-Cys-Tyr-{d-Trp}-Lys-Val-Cys-Trp-NH2 (Disulfide bridge: Cys2-Cys7)
Sequence shortening{d-Phe}-CY-{d-Trp}-KVCW-NH2 (Disulfide bridge: Cys2-Cys7)
SMILESCC(O)=O.O=C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N1)=O)C(C)C)=O)CCCCN)=O)CC2=CNC3=C2C=CC=C3)=O)CC4=CC=C(C=C4)O)=O)CSSC[C@H]1C(N[C@H](C(N)=O)CC5=CNC6=C5C=CC=C6)=O)[C@H](N)CC7=CC=CC=C7
SynonymsRC-160 acetate; BMY-41606 acetate
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This equation is commonly abbreviated as: C1V1 = C2V2

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GPCR/G Protein > Neurokinin Receptors