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Vapreotide diacetate

Catalog No.: A62143
Neurokinin Receptor Antagonist
Vapreotide diacetate is a neurokinin-1 (NK1) receptor antagonist with an IC50 of 330 nM. It exerts its biological activity by inhibiting NK1 receptor signaling, which plays a critical role in pain modulation, anxiety, and other neuropsychiatric conditions. This compound is employed in research applications targeting neurokinin signaling pathways, contributing to the exploration of therapeutic interventions for related disorders.
Vapreotide diacetate 936560-75-7 Neurokinin Receptor Antagonist
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Size Price Stock Qty
25mg
$1,275.00
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Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionVapreotide diacetate is a neurokinin-1 (NK1) receptor antagonist with an IC50 of 330 nM. It exerts its biological activity by inhibiting NK1 receptor signaling, which plays a critical role in pain modulation, anxiety, and other neuropsychiatric conditions. This compound is employed in research applications targeting neurokinin signaling pathways, contributing to the exploration of therapeutic interventions for related disorders.
Product Information
Catalog NumA62143
FormulaC61H78N12O13S2
Molecular Weight1251.47
CAS Number936560-75-7
Sequence{d-Phe}-Cys-Tyr-{d-Trp}-Lys-Val-Cys-Trp-NH2 (Disulfide bridge: Cys2-Cys7)
Sequence shortening{d-Phe}-CY-{d-Trp}-KVCW-NH2 (Disulfide bridge: Cys2-Cys7)
SMILESCC(O)=O.O=C([C@@H](NC([C@H](CSSC[C@H](NC([C@@H](NC([C@@H](NC1=O)CCCCN)=O)C(C)C)=O)C(N[C@H](C(N)=O)CC2=CNC3=CC=CC=C23)=O)NC([C@H](N)CC4=CC=CC=C4)=O)=O)CC5=CC=C(C=C5)O)N[C@@H]1CC6=CNC7=CC=CC=C67.CC(O)=O
SynonymsRC160 diacetate; BMY 41606 diacetate
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Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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This equation is commonly abbreviated as: C1V1 = C2V2

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GPCR/G Protein > Neurokinin Receptors