VU6005806

Catalog No.: A18488

M4 modulator

VU6005806

VU6005806 Chemical Structure

CAS NO. 2180914-37-6

VU6005806 (AZN-00016130) is a potent muscarnic acethylcholine receptor subtype 4 (M4) positive allosteric modulator (PAM), with EC50s of 94 nM, 28 nM, 87 nM and 68 nM for human, rat, dog and cyno M4, respectively. Used in the research of neuropsychiatric disorders.

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5 mg
$350.00
10 mg
$650.00
50 mg
$2,000.00
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Biological Activity

VU6005806 (AZN-00016130) is a potent muscarnic acethylcholine receptor subtype 4 (M4) positive allosteric modulator (PAM), with EC50s of 94 nM, 28 nM, 87 nM and 68 nM for human, rat, dog and cyno M4, respectively. Used in the research of neuropsychiatric disorders.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.76 mL 113.79 mL 227.58 mL
0.5 mM 4.55 mL 22.76 mL 45.52 mL
1 mM 2.28 mL 11.38 mL 22.76 mL
5 mM 0.46 mL 2.28 mL 4.55 mL

*The above data is based on the productmolecular weight 439.41. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18488
Actions Modulator
M. Wt 439.41
Formula C17H16F3N7O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2180914-37-6
Synonyms VU 6005806, VU-6005806, AZN00016130, AZN 00016130
SMILES NC1=C(C(NC2CN(C3=NC=C(C(F)(F)F)C=N3)C2)=O)SC4=NN=C(OC)C(C)=C41

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